Amide-to-chloroalkene substitution for overcoming intramolecular acyl transfer challenges in hexapeptidic neuromedin U receptor 2 agonists
掲載誌
Chem. Commun.
◎
巻,号,頁
60, 3563-3566
発行年
2024
発行月
2
著者
Shigenaga, A.*; Kyan, R.
4
論文題目
Theoretical study to gain fundamental insight into reaction mechanism of N-S acyl transfer of N-sulfanylethylanilide-based protein labeling reagent on protein surface
掲載誌
J. Pept. Sci. (Special Collection “Peptide Talents”)
Residue-selective C-H sulfenylation enabled by acid-activated S-acetamidomethyl cysteine sulfoxide with application to one-pot stapling and lipidation sequence
β,γ-trans-selective γ-butyrolactone formation via homoenolate cross-annulation of enals and aldehydes catalyzed by sterically hindered N-heterocyclic carbene
掲載誌
Tetrahedron
◎
巻,号,頁
91, 132191
発行年
2021
発行月
7
★
著者
Kyan, R.; Sato, K.; Mase, N.; Narumi, T.*
7
論文題目
Pendant Alkoxy Groups on N-Aryl Substitutions Drive the Efficiency of Imidazolylidene Catalysts for Homoenolate Annulation from Enal and Aldehyde
掲載誌
Angew. Chem. Int. Ed.
◎
巻,号,頁
59, 19031-19036
発行年
2020
発行月
★
著者
Ide, R.#; Kyan, R.#; Le, T. P.; Kitagawa, Y.; Sato, K.; Mase, N.; Narumi, T.* (#equally contribution)
8
論文題目
Chemoselective Umpolung of Enals for Asymmetric Homoenolate Cross-Annulation of Enals and Aldehydes Catalyzed by N-Heterocyclic Carbene